| Customization: | Available |
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| CAS No.: | 70918-53-5 |
| Formula: | N/a |
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(R)-1,4-benzodioxane-2-carboxylic acid, also known as (R)-baclofen carboxylic acid, is a chiral compound that serves as an intermediate in the synthesis of the pharmaceutical agent baclofen. Baclofen is a muscle relaxant primarily used to treat muscle spasms and spasticity resulting from conditions such as multiple sclerosis or spinal cord injuries. The (R)-enantiomer is the active form of the drug, highlighting the importance of stereochemistry in its therapeutic effects.
As a chemical intermediate, (R)-1,4-benzodioxane-2-carboxylic acid is involved in the synthesis of baclofen through a series of chemical reactions that ultimately yield the final product. The enantioselective synthesis of this compound is crucial to ensure that the final drug product contains the correct active isomer.
In the context of pharmaceutical development, the production of optically pure compounds like (R)-1,4-benzodioxane-2-carboxylic acid is essential to avoid the introduction of less active or potentially inactive enantiomers into the final medication. This is a key aspect of modern drug design and manufacturing, where the efficacy and safety of chiral drugs are closely tied to their stereochemical purity.
In summary, (R)-1,4-benzodioxane-2-carboxylic acid is a significant compound in the pharmaceutical industry due to its role in the production of the muscle relaxant baclofen. Its enantiomeric purity is critical for the effectiveness of the drug, emphasizing the importance of stereoselective synthesis in medicinal chemistry.
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