| Customization: | Available |
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| Transport Package: | Drum |
| Specification: | 99% |
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Cyproterone acetate is a synthetic steroid with strong anti-androgen properties and moderate progestogenic activity. It is used in the treatment of various conditions, including hormonal imbalances, prostate cancer, and as a component in some contraceptives.
Mechanism of Action: Cyproterone acetate works by blocking the effects of androgens (male sex hormones) in the body. It competitively inhibits the binding of androgens to their receptors, thereby reducing their activity. This results in a decrease in the production of sebum, which can be beneficial in treating conditions like acne and hirsutism. Additionally, it suppresses the secretion of luteinizing hormone (LH) and follicle-stimulating hormone (FSH), leading to a decrease in production.
Clinical Uses:
Pharmacokinetics: After oral administration, cyproterone acetate is rapidly absorbed and metabolized in the liver. Its bioavailability is high, and it has a long half-life, allowing for once or twice daily dosing.
Side Effects: Potential side effects include weight gain, mood changes, headache, dizziness, nausea, and breast tenderness. Long-term use may be associated with an increased risk of blood clots and liver function abnormalities.
Precautions: It is contraindicated in pregnancy and breastfeeding due to the potential for harm to the fetus or infant. It should also be used with caution in patients with a history of liver disease or blood clots.
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